Year | Title | Author(s) |
2019 |
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A
Journal Of Medicinal Chemistry |
Leaver, DJ Cleary, B Nguyen, N Priebbenow, DL Lagiakos, HR Sanchez, J Xue, L Huang, F Sun, YX Mujumdar, P Mudududdla, R Varghese, S Teguh, S Charman, SA White, KL Katneni, K Cuellar, M Strasser, JM Dahlin, JL Walters, MA Street, IP Monahan, BJ Jarman, KE Sabroux, HJ Falk, H Chung, MC Hermans, SJ Parker, MW Thomas, T Baell, JB |
2020 |
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents
Journal Of Medicinal Chemistry |
Priebbenow, DL Leaver, DJ Nguyen, N Cleary, B Lagiakos, HR Sanchez, J Xue, L Huang, F Sun, YX Mujumdar, P Mudududdla, R Varghese, S Teguh, S Charman, SA White, KL Shackleford, DM Katneni, K Cuellar, M Strasser, JM Dahlin, JL Walters, MA Street, IP Monahan, BJ Jarman, KE Sabroux, HJ Falk, H Chung, MC Hermans, SJ Downer, NL Parker, MW Voss, AK Thomas, T Baell, JB |
2021 |
Development of [F-18]MIPS15692, a radiotracer with in vitro proof-of-concept for the imaging of MER tyrosine kinase (MERTK) in neuroinflammatory disease
European Journal Of Medicinal Chemistry |
Wong, SW Vivash, L Mudududdla, R Nguyen, N Hermans, SJ Shackleford, DM Field, J Xue, L Aprico, A Hancock, NC Haskali, M Stashko, MA Frye, SV Wang, XD Binder, MD Ackermann, U Parker, MW Kilpatrick, TJ Baell, JB |