Year | Title | Author(s) |
2015 |
Crystal structure of human insulin-regulated aminopeptidase with specificity for cyclic peptides
Protein Science |
Hermans, SJ Ascher, DB Hancock, NC Holien, JK Michell, BJ Chai, SY Morton, CJ Parker, MW |
2015 |
Molecular basis for mid-region amyloid-beta capture by leading Alzheimer's disease immunotherapies
Scientific Reports |
Crespi, GAN Hermans, SJ Parker, MW Miles, LA |
2018 |
Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth
Nature |
Baell, JB Leaver, DJ Hermans, SJ Kelly, GL Brennan, MS Downer, NL Nguyen, N Wichmann, J Mcrae, HM Yang, YQ Cleary, B Lagiakos, HR Mieruszynski, S Pacini, G Vanyai, HK Bergamasco, MI May, RE Davey, BK Morgan, KJ Sealey, AJ Wang, BN Zamudio, N Wilcox, S Garnham, AL Sheikh, BN Aubrey, BJ Doggett, K Chung, MC de Silva, M Bentley, J Pilling, P Hattarki, M Dolezal, O Dennis, ML Falk, H Ren, B Charman, SA White, KL Rautela, J Newbold, A Hawkins, ED Johnstone, RW Huntington, ND Peat, TS Heath, JK Strasser, A Parker, MW Smyth, GK Street, IP Monahan, BJ Voss, AK Thomas, T |
2019 |
Small Molecule Binding to Alzheimer Risk Factor CD33 Promotes A beta Phagocytosis
Iscience |
Miles, LA Hermans, SJ Crespi, GAN Gooi, JH Doughty, L Nero, TL Markulic, J Ebneth, A Wroblowski, B Oehlrich, D Trabanco, AA Rives, ML Royaux, I Hancock, NC Parker, MW |
2019 |
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A
Journal Of Medicinal Chemistry |
Leaver, DJ Cleary, B Nguyen, N Priebbenow, DL Lagiakos, HR Sanchez, J Xue, L Huang, F Sun, YX Mujumdar, P Mudududdla, R Varghese, S Teguh, S Charman, SA White, KL Katneni, K Cuellar, M Strasser, JM Dahlin, JL Walters, MA Street, IP Monahan, BJ Jarman, KE Sabroux, HJ Falk, H Chung, MC Hermans, SJ Parker, MW Thomas, T Baell, JB |
2020 |
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents
Journal Of Medicinal Chemistry |
Priebbenow, DL Leaver, DJ Nguyen, N Cleary, B Lagiakos, HR Sanchez, J Xue, L Huang, F Sun, YX Mujumdar, P Mudududdla, R Varghese, S Teguh, S Charman, SA White, KL Shackleford, DM Katneni, K Cuellar, M Strasser, JM Dahlin, JL Walters, MA Street, IP Monahan, BJ Jarman, KE Sabroux, HJ Falk, H Chung, MC Hermans, SJ Downer, NL Parker, MW Voss, AK Thomas, T Baell, JB |
2021 |
Development of [F-18]MIPS15692, a radiotracer with in vitro proof-of-concept for the imaging of MER tyrosine kinase (MERTK) in neuroinflammatory disease
European Journal Of Medicinal Chemistry |
Wong, SW Vivash, L Mudududdla, R Nguyen, N Hermans, SJ Shackleford, DM Field, J Xue, L Aprico, A Hancock, NC Haskali, M Stashko, MA Frye, SV Wang, XD Binder, MD Ackermann, U Parker, MW Kilpatrick, TJ Baell, JB |